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| Drug Name | UNC0642 |
| Trade Name | |
| Synonyms | MP-IN-317 |
| Drug Descriptions |
UNC0642 (MP-IN-317) is a histone methyltransferase inhibitor that selectively inhibits EHMT2 (G9A) and EHMT1 (GLP), which may result in decreased methylation and potential cytotoxic effects against cancer cells (PMID: 24102134). |
| DrugClasses | EHMT2 Inhibitor 5 |
| CAS Registry Number | NA |
| NCIT ID | NA |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Afatinib + UNC0642 | Afatinib UNC0642 | 0 | 0 |
| UNC0642 | UNC0642 | 0 | 0 |