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Gene | CSF3R |
Variant | W791* |
Impact List | nonsense |
Protein Effect | gain of function |
Gene Variant Descriptions | CSF3R W791* results in a premature truncation of the Csf3r protein at amino acid 791 of 836 (UniProt.org). W791* results in increased cell surface Csf3r expression, hypersensitivity to G-CSF stimulation, elevated Stat5 activation, and is transforming in cell culture (PMID: 28439110). |
Associated Drug Resistance | |
Category Variants Paths |
CSF3R mutant CSF3R act mut CSF3R W791* |
Transcript | NM_000760.4 |
gDNA | chr1:g.36466496C>T |
cDNA | c.2372G>A |
Protein | p.W791* |
Source Database | RefSeq |
Genome Build | GRCh38/hg38 |
Transcript | gDNA | cDNA | Protein | Source Database | Genome Build |
---|---|---|---|---|---|
NM_000760.4 | chr1:g.36466496C>T | c.2372G>A | p.W791* | RefSeq | GRCh38/hg38 |
NM_000760.3 | chr1:g.36466496C>T | c.2372G>A | p.W791* | RefSeq | GRCh38/hg38 |
NM_000760 | chr1:g.36466496C>T | c.2372G>A | p.W791* | RefSeq | GRCh38/hg38 |
Molecular Profile | Indication/Tumor Type | Response Type | Therapy Name | Approval Status | Evidence Type | Efficacy Evidence | References |
---|---|---|---|---|---|---|---|
CSF3R W791* | hematologic cancer | predicted - sensitive | AZD1480 | Preclinical - Cell culture | Actionable | In a preclinical study, transformed hematologic cells expressing CSF3R W791* were sensitive to treatment with AZD1480 in culture, demonstrating decreased cell survival (PMID: 28031554). | 28031554 |
CSF3R W791* | hematologic cancer | predicted - resistant | Dasatinib | Preclinical - Cell culture | Actionable | In a preclinical study, transformed hematologic cells expressing CSF3R W791* demonstrated resistance to treatment with Sprycel (dasatinib) in culture (PMID: 28031554). | 28031554 |
CSF3R W791* | hematologic cancer | predicted - sensitive | Ruxolitinib | Preclinical - Cell culture | Actionable | In a preclinical study, transformed hematologic cells expressing CSF3R W791* were sensitive to treatment with Jakafi (ruxolitinib) in culture, demonstrating decreased cell survival (PMID: 28031554). | 28031554 |