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Gene | KIT |
Variant | K642E |
Impact List | missense |
Protein Effect | gain of function |
Gene Variant Descriptions | KIT K642E lies within the tyrosine kinase domain 1 (exon 13) of the Kit protein (PMID: 15990278). K642E results in constitutive phosphorylation of Kit and activation of downstream signaling (PMID: 15990278, PMID: 19802003), as well as transformation of cultured cells (PMID: 11073817). |
Associated Drug Resistance | |
Category Variants Paths |
KIT mutant KIT act mut KIT K642E KIT mutant KIT exon13 KIT K642E |
Transcript | NM_000222.3 |
gDNA | chr4:g.54728055A>G |
cDNA | c.1924A>G |
Protein | p.K642E |
Source Database | RefSeq |
Genome Build | GRCh38/hg38 |
Transcript | gDNA | cDNA | Protein | Source Database | Genome Build |
---|---|---|---|---|---|
NM_000222.2 | chr4:g.54728055A>G | c.1924A>G | p.K642E | RefSeq | GRCh38/hg38 |
NM_001385285.1 | chr4:g.54728055A>G | c.1924A>G | p.K642E | RefSeq | GRCh38/hg38 |
NM_000222 | chr4:g.54728055A>G | c.1924A>G | p.K642E | RefSeq | GRCh38/hg38 |
XM_017008178 | chr4:g.54728055A>G | c.1924A>G | p.K642E | RefSeq | GRCh38/hg38 |
NM_000222.3 | chr4:g.54728055A>G | c.1924A>G | p.K642E | RefSeq | GRCh38/hg38 |
XM_017008178.1 | chr4:g.54728055A>G | c.1924A>G | p.K642E | RefSeq | GRCh38/hg38 |
Molecular Profile | Protein Effect | Treatment Approaches |
---|---|---|
KIT K642E | gain of function | KIT Inhibitor |
KIT K642E KIT C809G KIT N822H | ||
KIT K642E KIT N822K | ||
KIT K642E KIT N822Y |