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Gene | FGFR1 |
Variant | V561M |
Impact List | missense |
Protein Effect | gain of function |
Gene Variant Descriptions | FGFR1 V561M lies within the protein kinase domain of the Fgfr1 protein (UniProt.org). V561M results in increased Fgfr1 autophosphorylation and has been shown to be associated with resistance to tyrosine kinase inhibitors (PMID: 25686244, PMID: 15157880, PMID: 28646488), and leads to increased Stat3 phosphorylation and STAT3-dependent gene expression, elevated expression of mesenchymal genes, and increased cell proliferation, migration, and anchorage-independent growth in culture (PMID: 30257990). |
Associated Drug Resistance | Y |
Category Variants Paths |
FGFR1 mutant FGFR1 act mut FGFR1 V561M |
Transcript | NM_023110.3 |
gDNA | chr8:g.38416043C>T |
cDNA | c.1681G>A |
Protein | p.V561M |
Source Database | RefSeq |
Genome Build | GRCh38/hg38 |
Transcript | gDNA | cDNA | Protein | Source Database | Genome Build |
---|---|---|---|---|---|
NM_023110.3 | chr8:g.38416043C>T | c.1681G>A | p.V561M | RefSeq | GRCh38/hg38 |
XM_006716303 | chr8:g.38416043C>T | c.1681G>A | p.V561M | RefSeq | GRCh38/hg38 |
NM_023110.2 | chr8:g.38416043C>T | c.1681G>A | p.V561M | RefSeq | GRCh38/hg38 |
XM_006716303.3 | chr8:g.38416043C>T | c.1681G>A | p.V561M | RefSeq | GRCh38/hg38 |
XM_017013221.1 | chr8:g.38416043C>T | c.1681G>A | p.V561M | RefSeq | GRCh38/hg38 |
XM_006716304.1 | chr8:g.38416043C>T | c.1681G>A | p.V561M | RefSeq | GRCh38/hg38 |
XM_006716304.2 | chr8:g.38416043C>T | c.1681G>A | p.V561M | RefSeq | GRCh38/hg38 |
XM_017013221 | chr8:g.38416043C>T | c.1681G>A | p.V561M | RefSeq | GRCh38/hg38 |
NM_023110 | chr8:g.38416043C>T | c.1681G>A | p.V561M | RefSeq | GRCh38/hg38 |
XM_006716303.4 | chr8:g.38416043C>T | c.1681G>A | p.V561M | RefSeq | GRCh38/hg38 |
XM_006716304 | chr8:g.38416043C>T | c.1681G>A | p.V561M | RefSeq | GRCh38/hg38 |
XM_017013221.2 | chr8:g.38416043C>T | c.1681G>A | p.V561M | RefSeq | GRCh38/hg38 |
Molecular Profile | Protein Effect | Treatment Approaches |
---|---|---|
FGFR1 V561M | gain of function | FGFR Inhibitor (Pan) FGFR1 Inhibitor |