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Gene | FLT3 |
Variant | R595_L601dup |
Impact List | duplication |
Protein Effect | gain of function |
Gene Variant Descriptions | FLT3 R595_L601dup (also referred to as FLT3 L601_K602insREYEYDL) indicates the insertion of seven duplicate amino acids, arginine (R)-595 through leucine(L)-601, in the juxtamembrane domain of the Flt3 protein (PMID: 11756186). R595_L601dup results in constitutive phosphorylation of Flt3, activation of Stat5 and Erk signaling, transformation of cells in culture, and induction of myeloproliferative disorder in mouse models (PMID: 18068628, PMID: 11756186). |
Associated Drug Resistance | |
Category Variants Paths |
FLT3 mutant FLT3 act mut FLT3 exon 14 ins FLT3 R595_L601dup FLT3 mutant FLT3 exon14 FLT3 exon 14 ins FLT3 R595_L601dup |
Transcript | NM_004119.3 |
gDNA | chr13:g.28034116_28034136 |
cDNA | c.1783_1803 |
Protein | p.R595_L601 |
Source Database | RefSeq |
Genome Build | GRCh38/hg38 |
Transcript | gDNA | cDNA | Protein | Source Database | Genome Build |
---|---|---|---|---|---|
NM_004119.3 | chr13:g.28034116_28034136 | c.1783_1803 | p.R595_L601 | RefSeq | GRCh38/hg38 |
NM_004119 | chr13:g.28034115_28034116insAAGGTCATACTCATACTCCCT | c.1804_1805insGGGAGTATGAGTATGACCTTA | p.R595_L601dup | RefSeq | GRCh38/hg38 |
Clinical Trial | Phase | Therapies | Title | Recruitment Status | Covered Countries | Other Countries |
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