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Gene | KIT |
Variant | C809G |
Impact List | missense |
Protein Effect | unknown |
Gene Variant Descriptions | KIT C809G lies within the protein kinase domain of the Kit protein (UniProt.org). C809G has been associated with secondary resistance to select KIT inhibitors (PMID: 16954519), but has not been biochemically characterized and therefore, its effect on Kit protein function is unknown (PubMed, Nov 2024). |
Associated Drug Resistance | Y |
Category Variants Paths |
KIT mutant KIT exon17 KIT C809G |
Transcript | NM_000222.3 |
gDNA | chr4:g.54733133T>G |
cDNA | c.2425T>G |
Protein | p.C809G |
Source Database | RefSeq |
Genome Build | GRCh38/hg38 |
Transcript | gDNA | cDNA | Protein | Source Database | Genome Build |
---|---|---|---|---|---|
NM_000222.3 | chr4:g.54733133T>G | c.2425T>G | p.C809G | RefSeq | GRCh38/hg38 |
NM_001385290.1 | chr4:g.54733133T>G | c.2425T>G | p.C809G | RefSeq | GRCh38/hg38 |
NM_000222 | chr4:g.54733133T>G | c.2425T>G | p.C809G | RefSeq | GRCh38/hg38 |
XM_005265741 | chr4:g.54733133T>G | c.2425T>G | p.C809G | RefSeq | GRCh38/hg38 |
NM_000222.2 | chr4:g.54733133T>G | c.2425T>G | p.C809G | RefSeq | GRCh38/hg38 |
XM_005265741.1 | chr4:g.54733133T>G | c.2425T>G | p.C809G | RefSeq | GRCh38/hg38 |
Molecular Profile | Indication/Tumor Type | Response Type | Therapy Name | Approval Status | Evidence Type | Efficacy Evidence | References |
---|---|---|---|---|---|---|---|
KIT C809G | Advanced Solid Tumor | predicted - resistant | Imatinib | Preclinical - Cell culture | Actionable | In a preclinical study, KIT C809G was resistant to inhibition of phosphorylation by Gleevec (imatinib) in cultured cells (PMID: 16954519). | 16954519 |