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Gene | PTEN |
Variant | L42R |
Impact List | missense |
Protein Effect | loss of function |
Gene Variant Descriptions | PTEN L42R lies within the phosphatase tensin-type domain of the Pten protein (UniProt.org). L42R demonstrates phosphatase activity comparable to wild-type Pten however, L42R results in reduced membrane localization of the Pten protein due to impaired binding with membrane lipids (PMID: 25448479, PMID: 25263454) and subsequently, is unable to prevent Akt signaling, cell proliferation, and cell migration and therefore, confers a loss of function to the Pten protein (PMID: 25263454). |
Associated Drug Resistance | |
Category Variants Paths |
PTEN mutant PTEN inact mut PTEN L42R |
Transcript | NM_000314.8 |
gDNA | chr10:g.87894070T>G |
cDNA | c.125T>G |
Protein | p.L42R |
Source Database | RefSeq |
Genome Build | GRCh38/hg38 |
Transcript | gDNA | cDNA | Protein | Source Database | Genome Build |
---|---|---|---|---|---|
NM_000314 | chr10:g.87894070T>G | c.125T>G | p.L42R | RefSeq | GRCh38/hg38 |
NM_001304717 | chr10:g.87864074T>G | c.125T>G | p.L42R | RefSeq | GRCh38/hg38 |
NM_001304717.2 | chr10:g.87864074T>G | c.125T>G | p.L42R | RefSeq | GRCh38/hg38 |
NM_001304717.5 | chr10:g.87864074T>G | c.125T>G | p.L42R | RefSeq | GRCh38/hg38 |
NM_000314.8 | chr10:g.87894070T>G | c.125T>G | p.L42R | RefSeq | GRCh38/hg38 |
NM_000314.6 | chr10:g.87894070T>G | c.125T>G | p.L42R | RefSeq | GRCh38/hg38 |
Molecular Profile | Protein Effect | Treatment Approaches |
---|---|---|
PTEN L42R | loss of function | Akt Inhibitor (Pan) Akt1 Inhibitor Akt2 Inhibitor PI3K Inhibitor (Pan) PIK3CB inhibitor |