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Gene | PIK3CA |
Variant | C971R |
Impact List | missense |
Protein Effect | gain of function - predicted |
Gene Variant Descriptions | PIK3CA C971R lies within the PI3K/PI4K domain of the Pik3ca protein (UniProt.org). C971R leads to Akt phosphorylation similar to wild-type Pik3ca (PMID: 34779417), but results in increased cell proliferation, viability, migration, and transformation ability compared to wild-type Pik3ca in several cell lines in culture (PMID: 29533785, PMID: 34779417), and in another study results in increased PI3K pathway signaling and moderate growth compared to control (PMID: 23619167), and therefore, is predicted to lead to a gain of Pik3ca protein function. |
Associated Drug Resistance | |
Category Variants Paths |
PIK3CA mutant PIK3CA act mut PIK3CA C971R PIK3CA mutant PIK3CA exon20 PIK3CA C971R |
Transcript | NM_006218.4 |
gDNA | chr3:g.179230351T>C |
cDNA | c.2911T>C |
Protein | p.C971R |
Source Database | RefSeq |
Genome Build | GRCh38/hg38 |
Transcript | gDNA | cDNA | Protein | Source Database | Genome Build |
---|---|---|---|---|---|
NM_006218.4 | chr3:g.179230351T>C | c.2911T>C | p.C971R | RefSeq | GRCh38/hg38 |
NM_006218 | chr3:g.179230351T>C | c.2911T>C | p.C971R | RefSeq | GRCh38/hg38 |
XM_011512894.2 | chr3:g.179230351T>C | c.2911T>C | p.C971R | RefSeq | GRCh38/hg38 |
XM_006713658.5 | chr3:g.179230351T>C | c.2911T>C | p.C971R | RefSeq | GRCh38/hg38 |
XM_006713658 | chr3:g.179230351T>C | c.2911T>C | p.C971R | RefSeq | GRCh38/hg38 |
XM_011512894 | chr3:g.179230351T>C | c.2911T>C | p.C971R | RefSeq | GRCh38/hg38 |
XM_006713658.4 | chr3:g.179230351T>C | c.2911T>C | p.C971R | RefSeq | GRCh38/hg38 |
NM_006218.3 | chr3:g.179230351T>C | c.2911T>C | p.C971R | RefSeq | GRCh38/hg38 |
Molecular Profile | Protein Effect | Treatment Approaches |
---|---|---|
PIK3CA C971R | gain of function - predicted | Akt Inhibitor (Pan) Akt1 Inhibitor Akt2 Inhibitor mTOR Inhibitor mTORC1 Inhibitor mTORC2 Inhibitor PI3K Inhibitor (Pan) PIK3CA inhibitor |