Missing content? – Request curation!
Request curation for specific Genes, Variants, or PubMed publications.
Have questions, comments, or suggestions? - Let us know!
Email us at : ckbsupport@genomenon.com
Gene | ROS1 |
Variant | D2113N |
Impact List | missense |
Protein Effect | gain of function |
Gene Variant Descriptions | ROS1 D2113N lies within the protein kinase domain of the Ros1 protein (UniProt.org). D2113N results in increased Ros1 activity, phosphorylation of Shp2 and Stat3, and colony formation in culture, and induces tumor formation in a mouse model (PMID: 37587872), and has been demonstrated to enhance resistance to ROS1 tyrosine kinase inhibitors with concurrent ROS1 G2032R in the context of a ROS1 fusion in culture (PMID: 26372962). |
Associated Drug Resistance | Y |
Category Variants Paths |
ROS1 mutant ROS1 act mut ROS1 D2113N |
Transcript | NM_002944.3 |
gDNA | chr6:g.117310178C>T |
cDNA | c.6337G>A |
Protein | p.D2113N |
Source Database | RefSeq |
Genome Build | GRCh38/hg38 |
Transcript | gDNA | cDNA | Protein | Source Database | Genome Build |
---|---|---|---|---|---|
NM_002944 | chr6:g.117310178C>T | c.6337G>A | p.D2113N | RefSeq | GRCh38/hg38 |
NM_002944.3 | chr6:g.117310178C>T | c.6337G>A | p.D2113N | RefSeq | GRCh38/hg38 |
NM_002944.2 | chr6:g.117310178C>T | c.6337G>A | p.D2113N | RefSeq | GRCh38/hg38 |
Molecular Profile | Indication/Tumor Type | Response Type | Therapy Name | Approval Status | Evidence Type | Efficacy Evidence | References |
---|