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Gene | JAK2 |
Variant | R938Q |
Impact List | missense |
Protein Effect | gain of function |
Gene Variant Descriptions | JAK2 R938Q lies within the protein kinase domain 2 of the Jak2 protein (UniProt.org). R938Q confers a gain of function to the Jak2 protein, as demonstrated by constitutive Stat5 signaling (PMID: 29025600), transformation of cultured cells (PMID: 24398328), and also displays resistance to Jak1/2 ATP-competitive inhibitors (PMID: 29025600). |
Associated Drug Resistance | Y |
Category Variants Paths |
JAK2 mutant JAK2 act mut JAK2 R938Q |
Transcript | NM_004972.4 |
gDNA | chr9:g.5090497G>A |
cDNA | c.2813G>A |
Protein | p.R938Q |
Source Database | RefSeq |
Genome Build | GRCh38/hg38 |
Transcript | gDNA | cDNA | Protein | Source Database | Genome Build |
---|---|---|---|---|---|
NM_004972 | chr9:g.5090497G>A | c.2813G>A | p.R938Q | RefSeq | GRCh38/hg38 |
NM_001322195.2 | chr9:g.5090497G>A | c.2813G>A | p.R938Q | RefSeq | GRCh38/hg38 |
NM_001322196 | chr9:g.5090497G>A | c.2813G>A | p.R938Q | RefSeq | GRCh38/hg38 |
NM_001322196.1 | chr9:g.5090497G>A | c.2813G>A | p.R938Q | RefSeq | GRCh38/hg38 |
NM_004972.3 | chr9:g.5090497G>A | c.2813G>A | p.R938Q | RefSeq | GRCh38/hg38 |
NM_001322195 | chr9:g.5090497G>A | c.2813G>A | p.R938Q | RefSeq | GRCh38/hg38 |
NM_004972.4 | chr9:g.5090497G>A | c.2813G>A | p.R938Q | RefSeq | GRCh38/hg38 |
NM_001322204 | chr9:g.5126414_5126415delAGinsCA | c.2812_2813delAGinsCA | p.R938Q | RefSeq | GRCh38/hg38 |
NM_001322196.2 | chr9:g.5090497G>A | c.2813G>A | p.R938Q | RefSeq | GRCh38/hg38 |
NM_001322194 | chr9:g.5090497G>A | c.2813G>A | p.R938Q | RefSeq | GRCh38/hg38 |
NM_001322204.1 | chr9:g.5126414_5126415delAGinsCA | c.2812_2813delAGinsCA | p.R938Q | RefSeq | GRCh38/hg38 |
NM_001322195.1 | chr9:g.5090497G>A | c.2813G>A | p.R938Q | RefSeq | GRCh38/hg38 |
NM_001322194.1 | chr9:g.5090497G>A | c.2813G>A | p.R938Q | RefSeq | GRCh38/hg38 |
NM_001322194.2 | chr9:g.5090497G>A | c.2813G>A | p.R938Q | RefSeq | GRCh38/hg38 |
NM_001322204.2 | chr9:g.5126414_5126415delAGinsCA | c.2812_2813delAGinsCA | p.R938Q | RefSeq | GRCh38/hg38 |
Molecular Profile | Indication/Tumor Type | Response Type | Therapy Name | Approval Status | Evidence Type | Efficacy Evidence | References |
---|---|---|---|---|---|---|---|
JAK2 R938Q | childhood B-cell acute lymphoblastic leukemia | resistant | Ruxolitinib | Preclinical - Patient cell culture | Actionable | In a preclinical study, bone marrow mononuclear cells from a pediatric B-cell acute lymphoblastic leukemia with an acquired Jak2 R938Q mutation were resistant to Jakafi (ruxolitinib) (PMID: 29025600). | 29025600 |