Missing content? – Request curation!
Request curation for specific Genes, Variants, or PubMed publications.
Have questions, comments, or suggestions? - Let us know!
Email us at : ckbsupport@genomenon.com
Gene | PIK3CA |
Variant | Q546K |
Impact List | missense |
Protein Effect | gain of function |
Gene Variant Descriptions | PIK3CA Q546K lies within the PIK helical domain of the Pik3ca protein (UniProt.org, PMID: 17376864). Q546K confers a gain of function to Pik3ca as indicated by constitutive phosphorylation of downstream targets Akt and S6, and is transforming in cell culture (PMID: 17376864, PMID: 29533785). |
Associated Drug Resistance | |
Category Variants Paths |
PIK3CA mutant PIK3CA act mut PIK3CA Q546K PIK3CA mutant PIK3CA exon10 PIK3CA Q546X PIK3CA Q546K |
Transcript | NM_006218.4 |
gDNA | chr3:g.179218306C>A |
cDNA | c.1636C>A |
Protein | p.Q546K |
Source Database | RefSeq |
Genome Build | GRCh38/hg38 |
Transcript | gDNA | cDNA | Protein | Source Database | Genome Build |
---|---|---|---|---|---|
XM_006713658 | chr3:g.179218306C>A | c.1636C>A | p.Q546K | RefSeq | GRCh38/hg38 |
XM_011512894 | chr3:g.179218306C>A | c.1636C>A | p.Q546K | RefSeq | GRCh38/hg38 |
NM_006218 | chr3:g.179218306C>A | c.1636C>A | p.Q546K | RefSeq | GRCh38/hg38 |
NM_006218.3 | chr3:g.179218306C>A | c.1636C>A | p.Q546K | RefSeq | GRCh38/hg38 |
XM_006713658.4 | chr3:g.179218306C>A | c.1636C>A | p.Q546K | RefSeq | GRCh38/hg38 |
XM_006713658.5 | chr3:g.179218306C>A | c.1636C>A | p.Q546K | RefSeq | GRCh38/hg38 |
NM_006218.4 | chr3:g.179218306C>A | c.1636C>A | p.Q546K | RefSeq | GRCh38/hg38 |
XM_011512894.2 | chr3:g.179218306C>A | c.1636C>A | p.Q546K | RefSeq | GRCh38/hg38 |
Molecular Profile | Protein Effect | Treatment Approaches |
---|---|---|
PIK3CA Q546K | gain of function | Akt Inhibitor (Pan) Akt1 Inhibitor Akt2 Inhibitor mTOR Inhibitor mTORC1 Inhibitor mTORC2 Inhibitor PI3K Inhibitor (Pan) PIK3CA inhibitor |