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Gene | PIK3CA |
Variant | Q546X |
Impact List | missense |
Protein Effect | unknown |
Gene Variant Descriptions | PIK3CA Q546X indicates any PIK3CA missense mutation that results in replacement of the glutamine (Q) at amino acid 546 by a different amino acid. |
Associated Drug Resistance | |
Category Variants Paths |
PIK3CA mutant PIK3CA exon10 PIK3CA Q546X |
Transcript | NM_006218.4 |
gDNA | chr3:g.179218306_179218308 |
cDNA | c.1636_1638 |
Protein | p.Q546 |
Source Database | RefSeq |
Genome Build | GRCh38/hg38 |
Transcript | gDNA | cDNA | Protein | Source Database | Genome Build |
---|---|---|---|---|---|
NM_006218.3 | chr3:g.179218306_179218308 | c.1636_1638 | p.Q546 | RefSeq | GRCh38/hg38 |
NM_006218.4 | chr3:g.179218306_179218308 | c.1636_1638 | p.Q546 | RefSeq | GRCh38/hg38 |
XM_006713658.5 | chr3:g.179218306_179218308 | c.1636_1638 | p.Q546 | RefSeq | GRCh38/hg38 |
XM_006713658.4 | chr3:g.179218306_179218308 | c.1636_1638 | p.Q546 | RefSeq | GRCh38/hg38 |
XM_011512894.2 | chr3:g.179218306_179218308 | c.1636_1638 | p.Q546 | RefSeq | GRCh38/hg38 |
Molecular Profile | Indication/Tumor Type | Response Type | Therapy Name | Approval Status | Evidence Type | Efficacy Evidence | References |
---|---|---|---|---|---|---|---|
PIK3CA Q546X | endometrial adenocarcinoma | no benefit | Copanlisib | Case Reports/Case Series | Actionable | In a Phase II (NRG-GY008) trial, Aliqopa (copanlisib) was well tolerated but demonstrated limited efficacy, resulted in 1 stable disease and 1 progressive disease in 2 patients with endometrioid adenocarcinoma harboring PIK3CA Q546 mutations, and stable disease in a patient with serous endometrial adenocarcinoma harboring a PIK3CA Q546 mutation (PMID: 31934607). | 31934607 |