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Gene | FGFR3 |
Variant | D641N |
Impact List | missense |
Protein Effect | gain of function - predicted |
Gene Variant Descriptions | FGFR3 D641N lies within the TK-2 domain of the Fgfr3 protein (PMID: 19287463). D641N results in proliferation similar to wild-type Fgfr3 in a competition assay and transformation activity similar to wild-type Fgfr3 in cultured cells (PMID: 34272467), but increased Fgfr3 autophosphorylation and substrate phosphorylation in culture (PMID: 26992226), and therefore, is predicted to lead to a gain of Fgfr3 protein function. |
Associated Drug Resistance | |
Category Variants Paths |
FGFR3 mutant FGFR3 act mut FGFR3 D641N |
Transcript | NM_000142.5 |
gDNA | chr4:g.1806135G>A |
cDNA | c.1921G>A |
Protein | p.D641N |
Source Database | RefSeq |
Genome Build | GRCh38/hg38 |
Transcript | gDNA | cDNA | Protein | Source Database | Genome Build |
---|---|---|---|---|---|
XM_006713873 | chr4:g.1806135G>A | c.1921G>A | p.D641N | RefSeq | GRCh38/hg38 |
NM_000142.4 | chr4:g.1806135G>A | c.1921G>A | p.D641N | RefSeq | GRCh38/hg38 |
NM_000142 | chr4:g.1806135G>A | c.1921G>A | p.D641N | RefSeq | GRCh38/hg38 |
XM_047449823.1 | chr4:g.1806135G>A | c.1921G>A | p.D641N | RefSeq | GRCh38/hg38 |
XM_006713873.2 | chr4:g.1806135G>A | c.1921G>A | p.D641N | RefSeq | GRCh38/hg38 |
XM_006713873.1 | chr4:g.1806135G>A | c.1921G>A | p.D641N | RefSeq | GRCh38/hg38 |
NM_000142.5 | chr4:g.1806135G>A | c.1921G>A | p.D641N | RefSeq | GRCh38/hg38 |
XM_047449824.1 | chr4:g.1806135G>A | c.1921G>A | p.D641N | RefSeq | GRCh38/hg38 |
Molecular Profile | Protein Effect | Treatment Approaches |
---|---|---|
FGFR3 D641N | gain of function - predicted | FGFR Inhibitor (Pan) FGFR3 Inhibitor |