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Gene | PIK3CA |
Variant | H1047Y |
Impact List | missense |
Protein Effect | gain of function |
Gene Variant Descriptions | PIK3CA H1047Y is a hotspot mutation that lies within the PI3K/PI4K domain of the Pik3ca protein (UniProt.org). H1047Y confers a gain of function on the Pik3ca protein as indicated by increased phosphorylation of Akt, activation of downstream signaling, and is transforming in cell culture (PMID: 17376864, PMID: 29533785). |
Associated Drug Resistance | |
Category Variants Paths |
PIK3CA mutant PIK3CA act mut PIK3CA H1047Y PIK3CA mutant PIK3CA exon21 PIK3CA H1047X PIK3CA H1047Y |
Transcript | NM_006218.4 |
gDNA | chr3:g.179234296C>T |
cDNA | c.3139C>T |
Protein | p.H1047Y |
Source Database | RefSeq |
Genome Build | GRCh38/hg38 |
Transcript | gDNA | cDNA | Protein | Source Database | Genome Build |
---|---|---|---|---|---|
NM_006218.3 | chr3:g.179234296C>T | c.3139C>T | p.H1047Y | RefSeq | GRCh38/hg38 |
XM_011512894 | chr3:g.179234296C>T | c.3139C>T | p.H1047Y | RefSeq | GRCh38/hg38 |
XM_006713658.4 | chr3:g.179234296C>T | c.3139C>T | p.H1047Y | RefSeq | GRCh38/hg38 |
XM_006713658 | chr3:g.179234296C>T | c.3139C>T | p.H1047Y | RefSeq | GRCh38/hg38 |
NM_006218.4 | chr3:g.179234296C>T | c.3139C>T | p.H1047Y | RefSeq | GRCh38/hg38 |
NM_006218 | chr3:g.179234296C>T | c.3139C>T | p.H1047Y | RefSeq | GRCh38/hg38 |
XM_006713658.5 | chr3:g.179234296C>T | c.3139C>T | p.H1047Y | RefSeq | GRCh38/hg38 |
XM_011512894.2 | chr3:g.179234296C>T | c.3139C>T | p.H1047Y | RefSeq | GRCh38/hg38 |
Molecular Profile | Protein Effect | Treatment Approaches |
---|---|---|
PIK3CA H1047Y | gain of function | Akt Inhibitor (Pan) Akt1 Inhibitor Akt2 Inhibitor mTOR Inhibitor mTORC1 Inhibitor mTORC2 Inhibitor PI3K Inhibitor (Pan) PIK3CA inhibitor |