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Gene | DNMT3A |
Variant | R882H |
Impact List | missense |
Protein Effect | loss of function |
Gene Variant Descriptions | DNMT3A R882H lies within the SAM-dependent MTase C5-type domain of the Dnmt3a protein (UniProt.org). R882H disrupts the tetramerization ability of the Dnmt3a protein, resulting in reduced DNA binding affinity and altered catalytic activity in in vitro assays (PMID: 22722925), disrupts Tp53 inhibition of methylation (PMID: 31640986), and results in hypomethylation, cytokine-independent growth, increased cell proliferation and impaired differentiation in cultured cells (PMID: 31164355, PMID: 32015320). |
Associated Drug Resistance | |
Category Variants Paths |
DNMT3A mutant DNMT3A inact mut DNMT3A R882H |
Transcript | NM_022552.5 |
gDNA | chr2:g.25234373C>T |
cDNA | c.2645G>A |
Protein | p.R882H |
Source Database | RefSeq |
Genome Build | GRCh38/hg38 |
Transcript | gDNA | cDNA | Protein | Source Database | Genome Build |
---|---|---|---|---|---|
XM_017003526.1 | chr2:g.25234373C>T | c.2645G>A | p.R882H | RefSeq | GRCh38/hg38 |
NM_022552 | chr2:g.25234373C>T | c.2645G>A | p.R882H | RefSeq | GRCh38/hg38 |
NM_175629 | chr2:g.25234373C>T | c.2645G>A | p.R882H | RefSeq | GRCh38/hg38 |
XM_017003526.2 | chr2:g.25234373C>T | c.2645G>A | p.R882H | RefSeq | GRCh38/hg38 |
NM_175629.2 | chr2:g.25234373C>T | c.2645G>A | p.R882H | RefSeq | GRCh38/hg38 |
XM_005264175.5 | chr2:g.25234373C>T | c.2645G>A | p.R882H | RefSeq | GRCh38/hg38 |
NM_175629.2 | chr2:g.25234373C>T | c.2645G>A | p.R882H | RefSeq | GRCh38/hg38 |
NM_022552.4 | chr2:g.25234373C>T | c.2645G>A | p.R882H | RefSeq | GRCh38/hg38 |
XM_005264175 | chr2:g.25234373C>T | c.2645G>A | p.R882H | RefSeq | GRCh38/hg38 |
XM_005264175.6 | chr2:g.25234373C>T | c.2645G>A | p.R882H | RefSeq | GRCh38/hg38 |
NM_022552.5 | chr2:g.25234373C>T | c.2645G>A | p.R882H | RefSeq | GRCh38/hg38 |
XM_017003526 | chr2:g.25234373C>T | c.2645G>A | p.R882H | RefSeq | GRCh38/hg38 |
Molecular Profile | Indication/Tumor Type | Response Type | Therapy Name | Approval Status | Evidence Type | Efficacy Evidence | References |
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