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Gene | FLT3 |
Variant | C790S |
Impact List | missense |
Protein Effect | gain of function - predicted |
Gene Variant Descriptions | FLT3 C790S lies within the protein kinase domain of the Flt3 protein (UniProt.org). C790S does not alter kinase activity, dimerization, cytokine-independent growth, or phosphorylation of Flt3 or Erk but results in increased colony formation and phosphorylation of Stat5 in the context of FLT3 internal tandem duplication (FLT3-ITD) and results in increased kinase activity compared to wild-type Flt3 in cultured cells (PMID: 31606550), and therefore, is predicted to lead to a gain of Flt3 protein function. |
Associated Drug Resistance | |
Category Variants Paths |
FLT3 mutant FLT3 act mut FLT3 C790S FLT3 mutant FLT3 exon19 FLT3 C790S |
Transcript | NM_004119.3 |
gDNA | chr13:g.28023400A>T |
cDNA | c.2368T>A |
Protein | p.C790S |
Source Database | RefSeq |
Genome Build | GRCh38/hg38 |
Transcript | gDNA | cDNA | Protein | Source Database | Genome Build |
---|---|---|---|---|---|
XM_011535018.3 | chr13:g.28004141A>T | c.2368T>A | p.C790S | RefSeq | GRCh38/hg38 |
NM_004119.3 | chr13:g.28023400A>T | c.2368T>A | p.C790S | RefSeq | GRCh38/hg38 |
XM_047430216.1 | chr13:g.28004141A>T | c.2368T>A | p.C790S | RefSeq | GRCh38/hg38 |
NM_004119.2 | chr13:g.28023400A>T | c.2368T>A | p.C790S | RefSeq | GRCh38/hg38 |
Molecular Profile | Indication/Tumor Type | Response Type | Therapy Name | Approval Status | Evidence Type | Efficacy Evidence | References |
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