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Gene | FLT3 |
Variant | F590_D593delinsGP |
Impact List | indel |
Protein Effect | unknown |
Gene Variant Descriptions | FLT3 F590_D593delinsGP results in a deletion of four amino acids in the juxtamembrane domain of the Flt3 protein from amino acids 590 to 593, combined with the insertion of a glycine (G) and a proline (P) at the same site (PMID: 37246158). F590_D593delinsGP results in Flt3 phosphorylation similar to wild-type Flt3 in culture (PMID: 37246158), but has not been fully biochemically characterized and therefore, its effect on Flt3 protein function is unknown. |
Associated Drug Resistance | |
Category Variants Paths |
FLT3 mutant FLT3 exon14 FLT3 F590_D593delinsGP |
Transcript | NM_004119.2 |
gDNA | chr13:g.28034140_28034151delinsAGGACC |
cDNA | c.1768_1779delinsGGTCCT |
Protein | p.F590_D593delinsGP |
Source Database | RefSeq |
Genome Build | GRCh38/hg38 |
Transcript | gDNA | cDNA | Protein | Source Database | Genome Build |
---|---|---|---|---|---|
NM_004119.2 | chr13:g.28034140_28034151delinsAGGACC | c.1768_1779delinsGGTCCT | p.F590_D593delinsGP | RefSeq | GRCh38/hg38 |
Molecular Profile | Indication/Tumor Type | Response Type | Therapy Name | Approval Status | Evidence Type | Efficacy Evidence | References |
---|---|---|---|---|---|---|---|
FLT3 F590_D593delinsGP | hematologic cancer | predicted - sensitive | Quizartinib | Preclinical - Biochemical | Actionable | In a preclinical study, Vanflyta (quizartinib) inhibited Flt3 phosphorylation in cells expressing FLT3 F590_D593delinsGP in culture (PMID: 37246158). | 37246158 |
FLT3 F590_D593delinsGP | hematologic cancer | predicted - sensitive | Sorafenib | Preclinical - Biochemical | Actionable | In a preclinical study, Nexavar (sorafenib) inhibited Flt3 phosphorylation in cells expressing FLT3 F590_D593delinsGP in culture (PMID: 37246158). | 37246158 |