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Gene | CHEK2 |
Variant | R474H |
Impact List | missense |
Protein Effect | loss of function |
Gene Variant Descriptions | CHEK2 R474H lies within the protein kinase domain of the Chek2 protein (UniProt.org). R474H results in decreased Chek2 protein stability in culture (PMID: 34903604), and results in a loss of Kap1 phosphorylation at serine (S)-473 compared to wild-type Chek2 in culture and in vitro assays (PMID: 31050813, PMID: 34903604). |
Associated Drug Resistance | |
Category Variants Paths |
CHEK2 mutant CHEK2 inact mut CHEK2 R474H |
Transcript | NM_007194.4 |
gDNA | chr22:g.28694072C>T |
cDNA | c.1421G>A |
Protein | p.R474H |
Source Database | RefSeq |
Genome Build | GRCh38/hg38 |
Transcript | gDNA | cDNA | Protein | Source Database | Genome Build |
---|---|---|---|---|---|
NM_001005735.1 | chr22:g.28695209_28695211delAGGinsCAT | c.1420_1422delAGGinsCAT | p.R474H | RefSeq | GRCh38/hg38 |
NM_007194.3 | chr22:g.28694072C>T | c.1421G>A | p.R474H | RefSeq | GRCh38/hg38 |
XM_024452149.1 | chr22:g.28689198_28689200delAGAinsCAT | c.1420_1422delAGAinsCAT | p.R474H | RefSeq | GRCh38/hg38 |
NM_007194.4 | chr22:g.28694072C>T | c.1421G>A | p.R474H | RefSeq | GRCh38/hg38 |
NM_001005735.2 | chr22:g.28695209_28695211delAGGinsCAT | c.1420_1422delAGGinsCAT | p.R474H | RefSeq | GRCh38/hg38 |
NM_007194 | chr22:g.28694072C>T | c.1421G>A | p.R474H | RefSeq | GRCh38/hg38 |
NM_001005735 | chr22:g.28695209_28695211delCCTinsATG | c.1420_1422delAGGinsCAT | p.R474H | RefSeq | GRCh38/hg38 |
XM_024452149.2 | chr22:g.28689198_28689200delAGAinsCAT | c.1420_1422delAGAinsCAT | p.R474H | RefSeq | GRCh38/hg38 |
Molecular Profile | Protein Effect | Treatment Approaches |
---|---|---|
CHEK2 R474H | loss of function | Olaparib |