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Gene | FGFR2 |
Variant | M538I |
Impact List | missense |
Protein Effect | gain of function |
Gene Variant Descriptions | FGFR2 M538I (corresponds to M537I in the canonical isoform) lies within the protein kinase domain of the Fgfr2 protein (UniProt.org). M538I confers a gain of function to the Fgfr2 protein as demonstrated by increased Fgfr2 kinase activity (PMID: 32723837, PMID: 23908597) and enhanced cell proliferation in the presence of ligand in cell culture (PMID: 23908597), and has been associated with decreased sensitivity to some FGFR inhibitors (PMID: 23908597). |
Associated Drug Resistance | |
Category Variants Paths |
FGFR2 mutant FGFR2 act mut FGFR2 M538I |
Transcript | NM_000141.5 |
gDNA | chr10:g.121498553C>G |
cDNA | c.1614G>C |
Protein | p.M538I |
Source Database | RefSeq |
Genome Build | GRCh38/hg38 |
Transcript | gDNA | cDNA | Protein | Source Database | Genome Build |
---|---|---|---|---|---|
NM_001320658 | chr10:g.121498547C>G | c.1614G>C | p.M538I | RefSeq | GRCh38/hg38 |
NM_001144913.1 | chr10:g.121498556C>G | c.1614G>C | p.M538I | RefSeq | GRCh38/hg38 |
NM_001144913.1 | chr10:g.121498556C>G | c.1614G>C | p.M538I | RefSeq | GRCh38/hg38 |
XM_006717710.4 | chr10:g.121500833C>G | c.1614G>C | p.M538I | RefSeq | GRCh38/hg38 |
NM_000141 | chr10:g.121498553C>G | c.1614G>C | p.M538I | RefSeq | GRCh38/hg38 |
XM_006717710.5 | chr10:g.121500833C>G | c.1614G>C | p.M538I | RefSeq | GRCh38/hg38 |
NM_000141.5 | chr10:g.121498553C>G | c.1614G>C | p.M538I | RefSeq | GRCh38/hg38 |
NM_022970 | chr10:g.121498556C>G | c.1614G>C | p.M538I | RefSeq | GRCh38/hg38 |
NM_001144913 | chr10:g.121498556C>G | c.1614G>C | p.M538I | RefSeq | GRCh38/hg38 |
NM_000141.4 | chr10:g.121498553C>G | c.1614G>C | p.M538I | RefSeq | GRCh38/hg38 |
XM_006717710 | chr10:g.121500833C>G | c.1614G>C | p.M538I | RefSeq | GRCh38/hg38 |
NM_001320658.1 | chr10:g.121498547C>G | c.1614G>C | p.M538I | RefSeq | GRCh38/hg38 |
NM_022970.4 | chr10:g.121498556C>G | c.1614G>C | p.M538I | RefSeq | GRCh38/hg38 |
NM_001320658.2 | chr10:g.121498547C>G | c.1614G>C | p.M538I | RefSeq | GRCh38/hg38 |
NM_022970.3 | chr10:g.121498556C>G | c.1614G>C | p.M538I | RefSeq | GRCh38/hg38 |
Molecular Profile | Protein Effect | Treatment Approaches |
---|---|---|
FGFR2 M538I | gain of function | FGFR Inhibitor (Pan) FGFR2 Inhibitor |
FGFR2 fusion FGFR2 M538I |