Lirafugratinib
Drug Detail
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| Drug Name | Lirafugratinib |
| Trade Name | |
| Synonyms | RLY4008|RLY 4008|RLY-4008 |
| Drug Descriptions |
Lirafugratinib binds to and inhibits FGFR2, selectively targeting primary oncogenic FGFR2 mutations and leads to decreased FGFR2-dependent signaling, potentially resulting in inhibition of tumor cell proliferation (NCI Drug Dictionary; Journal of Clinical Oncology 39, no. 15_suppl). |
| DrugClasses | FGFR2 Inhibitor 24 |
| CAS Registry Number | 2549174-42-5 |
| NCIT ID | C174208 |
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| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Lirafugratinib | Lirafugratinib | 16 | 1 |
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