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| Drug Name | BLU-451 |
| Trade Name | |
| Synonyms | BLU451|BLU 451|LNG-451|LNG451|LNG 451 |
| Drug Descriptions |
BLU-451 is a blood-brain-barrier penetrant, mutant-selective, EGFR inhibitor with activity against exon 20 insertions, which blocks downstream signaling potentially resulting in decreased tumor growth (NCI Drug Dictionary). |
| DrugClasses | EGFR Exon 20 Insertion Inhibitor 13 |
| CAS Registry Number | NA |
| NCIT ID | C187042 |
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| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| BLU-451 | BLU-451 | 0 | 1 |
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