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Drug Name | HSK29116 |
Trade Name | |
Synonyms | HSK-29116|HSK 29116 |
Drug Descriptions |
HSK29116 is a proteolysis-targeted chimera (PROTAC) that binds to Bruton's tyrosine kinase (BTK) and targets it for degradation, potentially leading to growth inhibition in BTK-expressing tumor cells (NCI Drug Dictionary). |
DrugClasses | BTK inhibitor 38 |
CAS Registry Number | NA |
NCIT ID | C180676 |
Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
---|---|---|---|
HSK29116 | HSK29116 | 0 | 1 |