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| Drug Name | KSQ-4279 |
| Trade Name | |
| Synonyms | KSQ 4279|KSQ4279 |
| Drug Descriptions |
KSQ-4279 inhibits Usp1 deubiquitinase activity, potentially leading to apoptosis and decreased tumor growth (PMID: 39402989). |
| DrugClasses | USP1 inhibitor 7 |
| CAS Registry Number | 2446480-97-1 |
| NCIT ID | C185613 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| KSQ-4279 | KSQ-4279 | 0 | 1 |
| KSQ-4279 + Olaparib | KSQ-4279 Olaparib | 0 | 0 |
| KSQ-4279 + Saruparib | KSQ-4279 Saruparib | 0 | 0 |