Missing content? – Request curation!
Request curation for specific Genes, Variants, or PubMed publications.
Have questions, comments, or suggestions? - Let us know!
Email us at : ckbsupport@genomenon.com
| Drug Name | FCN-159 |
| Trade Name | |
| Synonyms | FCN159|FCN 159 |
| Drug Descriptions |
FCN-159 inhibits MAP2K1/2 (MEK1/2), potentially resulting in reduced proliferation and increased cell cycle arrest and apoptosis in tumor cells, and inhibition of tumor growth (Cancer Res 2020;80(16 Suppl):Abstract nr 1951). |
| DrugClasses | MEK1 Inhibitor 27 MEK2 Inhibitor 25 |
| CAS Registry Number | NA |
| NCIT ID | C172382 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| FCN-159 | FCN-159 | 3 | 1 |