KT-253
Drug Detail
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| Drug Name | KT-253 |
| Trade Name | |
| Synonyms | KT 253|KT253 |
| Drug Descriptions |
KT-253 is a degrader of MDM2, which reduces TP53-dependent increase in MDM2 protein levels and potentially induces apoptosis in tumor cells and inhibits tumor growth (Blood (2022) 140 (Supplement 1): 6239-6240). |
| DrugClasses | MDM2 Inhibitor 23 |
| CAS Registry Number | NA |
| NCIT ID | NA |
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| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| KT-253 | KT-253 | 0 | 1 |
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