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| Drug Name | GSK4524101 |
| Trade Name | |
| Synonyms | GSK 4524101|GSK-4524101 |
| Drug Descriptions |
GSK4524101 inhibits DNA polymerase theta, which may prevent the repair of DNA-double stranded breaks, resulting in decreased tumor cell proliferation (Cancer Res (2024) 84 (7_Supplement): CT169, NCI Drug Dictionary). |
| DrugClasses | |
| CAS Registry Number | NA |
| NCIT ID | C201946 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| GSK4524101 | GSK4524101 | 0 | 1 |
| GSK4524101 + Niraparib | GSK4524101 Niraparib | 0 | 1 |