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| Drug Name | 177Lu-FF58 |
| Trade Name | |
| Synonyms | 177LuFF58|[177Lu]-FF58|Lutetium Lu 177 FF58 |
| Drug Descriptions |
177Lu-FF58 is a radioconjugate comprising a non-RGD small molecule that targets integrins alphaVbeta3 and alphaVbeta5 conjugated to the radionuclide lutetium-177, which delivers beta radiation to tumor cells expressing integrin alphaVbeta3 or alphaVbeta5, potentially resulting in antitumor activity (NCI Drug Dictionary). |
| DrugClasses | |
| CAS Registry Number | NA |
| NCIT ID | C205213 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| 177Lu-FF58 | 177Lu-FF58 | 0 | 1 |