SHR2554
Drug Detail
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| Drug Name | SHR2554 |
| Trade Name | |
| Synonyms | SHR-2554|SHR 2554|TLN254|TLN-254|TLN 254|Zeprumetostat |
| Drug Descriptions |
SHR2554 inhibits wild-type and mutant EZH2, which potentially decreases intracellular H3K27me3 and reduces tumor growth (PMID: 38190117). |
| DrugClasses | EZH2 inhibitor 20 |
| CAS Registry Number | 2098545-98-1 |
| NCIT ID | C158742 |
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| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| SHR2554 | SHR2554 | 0 | 1 |
| SHR2554 + TLN-121 | SHR2554 TLN-121 | 0 | 1 |
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