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| Drug Name | ASP4396 |
| Trade Name | |
| Synonyms | ASP-4396|ASP 4396 |
| Drug Descriptions |
ASP4396 comprises a E3 ubiquitin ligase-binding moiety linked to a moiety targeting KRAS G12D, which potentially targets KRAS G12D for proteasomal degradation, resulting in decreased growth of KRAS G12D-expressing tumor cells (NCI Drug Dictionary). |
| DrugClasses | KRAS G12D Inhibitor 25 |
| CAS Registry Number | NA |
| NCIT ID | C212079 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| ASP4396 | ASP4396 | 0 | 1 |