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Drug Name OPN-6602
Trade Name
Synonyms OPN6602|OPN 6602
Drug Descriptions

OPN-6602 is a small molecule inhibitor of EP300 (p300) and CBP (CREBBP), which downregulates IRF4 and MYC, potentially inhibiting tumor growth (Cancer Res (2024) 84 (6_Supplement): 660).

DrugClasses CBP/p300 inhibitor 13
CAS Registry Number
NCIT ID

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Therapy Name Drugs Efficacy Evidence Clinical Trials
Dexamethasone + OPN-6602 Dexamethasone OPN-6602 0 1
Lenalidomide + OPN-6602 Lenalidomide OPN-6602 0 0
OPN-6602 OPN-6602 0 1


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