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| Drug Name | YH42946 |
| Trade Name | |
| Synonyms | YH-42946|YH 42946 |
| Drug Descriptions |
YH42946 is a small molecule EGFR inhibitor with selectivity for EGFR exon 20 insertion mutations, which potentially inhibits tumor cell viability (Cancer Res (2025) 85 (8_Supplement_1): 5604). |
| DrugClasses | EGFR Exon 20 Insertion Inhibitor 15 |
| CAS Registry Number | NA |
| NCIT ID | NA |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| YH42946 | YH42946 | 0 | 1 |