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Drug Name | (R)-9bMS |
Trade Name | |
Synonyms | (R) 9bMS|(R)9bMS|Mahatinib |
Drug Descriptions |
(R)-9bMS inhibits TNK2 (ACK1) and suppresses AR gene expression, potentially leading to decreased tumor cell proliferation and inhibition of tumor growth (PMID: 36861798, PMID: 27902967, PMID: 28609657). |
DrugClasses | TNK2 Inhibitor 7 |
CAS Registry Number | 1655527-68-6 |
NCIT ID | NA |
Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
---|---|---|---|
(R)-9bMS | (R)-9bMS | 0 | 1 |