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| Drug Name | 177Lu-FAP-2286 |
| Trade Name | |
| Synonyms | 177-FAP-2286|FAP-2286|FAP 2286|Lutetium Lu 177-FAP-2286 |
| Drug Descriptions |
177Lu-FAP-2286 is a radioconjugate comprising a FAP-binding cyclic peptide linked to a DOTA chelator labeled with the radionuclide Lutetium-177, which potentially inhibits growth of FAP-expressing tumors (PMID: 35608703). |
| DrugClasses | |
| CAS Registry Number | NA |
| NCIT ID | C180806 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| 177Lu-FAP-2286 | 177Lu-FAP-2286 | 0 | 1 |