Missing content? – Request curation!
Request curation for specific Genes, Variants, or PubMed publications.
Have questions, comments, or suggestions? - Let us know!
Email us at : ckbsupport@genomenon.com
| Drug Name | FORX-428 |
| Trade Name | |
| Synonyms | FORX 428|FORX428 |
| Drug Descriptions |
FORX-428 inhibits poly (ADP-ribose) glycohydrolase (PARG) and leads to increased sensitivity to DNA damage and replication stress, which may result in anti-tumor activity (Mol Cancer Ther (2025) 24 (10_Supplement): B022). |
| DrugClasses | |
| CAS Registry Number | NA |
| NCIT ID | NA |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| FORX-428 | FORX-428 | 0 | 1 |