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| Drug Name | BMS-777607 |
| Trade Name | |
| Synonyms | ASLAN002|BMS777607|BMS 777607 |
| Drug Descriptions |
BMS-777607 (ASLAN002) is a small molecule that inhibits MET, MST1R (RON), TYRO3, and AXL, resulting in decreased downstream pathway activation, potentially resulting in decreased tumor cell growth and metastasis (PMID: 19260711, PMID: 20515943, PMID: 24233399, PMID: 26555154). |
| DrugClasses | AXL Inhibitor 30 MET Inhibitor 59 RON Inhibitor 11 TYRO3 Inhibitor 7 |
| CAS Registry Number | 1025720-94-8 |
| NCIT ID | C74060 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| BMS-777607 | BMS-777607 | 0 | 0 |
| BMS-777607 + Buparlisib | BMS-777607 Buparlisib | 0 | 0 |
| BMS-777607 + Trametinib | BMS-777607 Trametinib | 0 | 0 |