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Drug Name | GSK2126458 |
Trade Name | |
Synonyms | GSK458|Omipalisib |
Drug Descriptions |
Omipalisib (GSK2126458) is a dual pan-PI3K and mTOR inhibitor, which blocks PI3K/AKT signaling to prevent cell proliferation (PMID: 24900173, PMID: 32382996). |
DrugClasses | mTOR Inhibitor 51 PI3K Inhibitor (Pan) 42 |
CAS Registry Number | 1086062-66-9 |
NCIT ID | C88270 |