Masitinib
Drug Detail
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| Drug Name | Masitinib |
| Trade Name | |
| Synonyms | AB1010 |
| Drug Descriptions |
Masitinib (AB1010) inhibits several receptor tyrosine kinases including c-KIT, PDGFR, and LYN, which may result in inhibition of cell proliferation (PMID: 19789626, PMID: 29638149). |
| DrugClasses | KIT Inhibitor 57 LYN Inhibitor 4 PDGFR Inhibitor (Pan) 30 |
| CAS Registry Number | 790299-79-5 |
| NCIT ID | C79910 |
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| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Docetaxel + Masitinib + Prednisone | Docetaxel Masitinib Prednisone | 0 | 1 |
| Gemcitabine + Masitinib | Gemcitabine Masitinib | 0 | 0 |
| Masitinib | Masitinib | 0 | 5 |
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