Missing content? – Request curation!
Request curation for specific Genes, Variants, or PubMed publications.
Have questions, comments, or suggestions? - Let us know!
Email us at : ckbsupport@genomenon.com
| Drug Name | Belizatinib |
| Trade Name | |
| Synonyms | TSR-011 |
| Drug Descriptions |
Belizatinib (TSR-011) binds to ALK and TRK kinases and inhibits downstream signaling, which may result in decreased proliferation of ALK/TRK expressing tumor cells (PMID: 26753004, PMID: 31217479). |
| DrugClasses | ALK Inhibitor 33 Trk Receptor Inhibitor (Pan) 33 |
| CAS Registry Number | 1357920-84-3 |
| NCIT ID | C169804 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Belizatinib | Belizatinib | 6 | 1 |