Epertinib
Drug Detail
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| Drug Name | Epertinib |
| Trade Name | |
| Synonyms | S-222611|S222611|S222611 |
| Drug Descriptions |
Epertinib (S-222611) is a dual inhibitor of EGFR and ERBB2 (HER2), leading to decreased kinase activity and potentially inhibiting growth of tumors expressing EGFR or ERBB2 (HER2) (PMID: 24837299, PMID: 30196106, PMID: 31892325). |
| DrugClasses | EGFR Inhibitor (Pan) 63 HER2 Inhibitor 44 |
| CAS Registry Number | 908305-13-5 |
| NCIT ID | C166884 |
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| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Epertinib | Epertinib | 0 | 0 |
| Epertinib + Trastuzumab | Epertinib Trastuzumab | 0 | 0 |
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