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| Drug Name | SAR260301 |
| Trade Name | |
| Synonyms | SAR 260301|SAR-260301 |
| Drug Descriptions |
SAR260301 is PI3K beta-selective inhibitor, which has been demonstrated to inhibit tumor growth in xenograft models (PMID: 24387221, PMID: 28976556). |
| DrugClasses | PIK3CB inhibitor 8 |
| CAS Registry Number | 1260612-13-2 |
| NCIT ID | C116882 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| SAR260301 | SAR260301 | 4 | 1 |
| SAR260301 + Selumetinib | SAR260301 Selumetinib | 1 | 0 |
| SAR260301 + Vemurafenib | SAR260301 Vemurafenib | 1 | 1 |