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| Drug Name | CCT241533 |
| Trade Name | |
| Synonyms | CCT 241533|CCT-241533 |
| Drug Descriptions |
CCT241533 is an ATP-competitive inhibitor of CHK2, which enhances PARP inhibitor efficacy in cells lacking functional TP53 (PMID: 21239475). |
| DrugClasses | CHK2 Inhibitor 7 |
| CAS Registry Number | 1262849-73-9 |
| NCIT ID | NA |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| CCT241533 | CCT241533 | 0 | 0 |
| CCT241533 + Olaparib | CCT241533 Olaparib | 0 | 0 |
| CCT241533 + Rucaparib | CCT241533 Rucaparib | 0 | 0 |