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| Drug Name | Ilginatinib |
| Trade Name | |
| Synonyms | NS-018 |
| Drug Descriptions |
Ilginatinib (NS-018) inhibits JAK2, including JAK2 V617F, as well as SRC family members, including SRC, FYN, and YES, potentially leading to decreased cell proliferation (PMID: 24413068, PMID: 22829185, PMID: 29941953). |
| DrugClasses | JAK2 Inhibitor - ATP competitive 15 SRC Inhibitor 31 YES Inhibitor 3 |
| CAS Registry Number | 1239358-86-1 |
| NCIT ID | C98109 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Ilginatinib | Ilginatinib | 2 | 1 |