MK-8242
Drug Detail
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| Drug Name | MK-8242 |
| Trade Name | |
| Synonyms | SCH 900242 |
| Drug Descriptions |
MK-8242 binds MDM2 and prevents its interaction with p53, thereby inhibiting degradation of p53 and potentially resulting in increased tumor cell apoptosis (PMID: 30253242). |
| DrugClasses | MDM2 Inhibitor 23 |
| CAS Registry Number | NA |
| NCIT ID | C116867 |
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| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| MK-8242 | MK-8242 | 2 | 0 |
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