MK8033
Drug Detail
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| Drug Name | MK8033 |
| Trade Name | |
| Synonyms | MK-8033|HQP8361|HQP 8361|HQP-8361|MK 8033 |
| Drug Descriptions |
MK8033 is an inhibitor of MET and MST1R (RON) that suppresses mTOR signaling, potentially resulting in reduced survival and colony formation, increased apoptosis, and inhibition of tumor growth (PMID: 23792360, PMID: 33163272). |
| DrugClasses | MET Inhibitor 59 RON Inhibitor 11 |
| CAS Registry Number | 1196681-38-5 |
| NCIT ID | C116866 |
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| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| MK8033 | MK8033 | 0 | 0 |
| MK8033 + Osimertinib | MK8033 Osimertinib | 0 | 0 |
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