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| Drug Name | TP-3654 |
| Trade Name | |
| Synonyms | SGI-9481|SGI9481|TP3654 |
| Drug Descriptions |
TP-3654 (SGI-9481) is an inhibitor of PIM1, PIM2, PIM3, and moderately inhibits FLT3, which may result in anti-tumor activity (PMID: 24953177). |
| DrugClasses | FLT3 Inhibitor 69 PIM Inhibitor (Pan) 10 |
| CAS Registry Number | 1361951-15-6 |
| NCIT ID | C160203 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| TP-3654 | TP-3654 | 0 | 2 |