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| Drug Name | Ch282-5 |
| Trade Name | |
| Synonyms | |
| Drug Descriptions |
Ch282-5 is a gossypol derivative that binds to and inhibits BCL2, family proteins, resulting in decreased tumor cell growth and increased sensitivity to chemotherapeutic agents (PMID: 26515494, PMID: 29885833). |
| DrugClasses | BCL2 Family Inhibitor 6 |
| CAS Registry Number | NA |
| NCIT ID | NA |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Ch282-5 | Ch282-5 | 0 | 0 |
| Ch282-5 + Oxaliplatin | Ch282-5 Oxaliplatin | 0 | 0 |