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| Drug Name | THZ1 |
| Trade Name | |
| Synonyms | HY-80013|THZ-1 |
| Drug Descriptions |
THZ1 is a covalent Cdk7 inhibitor that inhibits tumor cell proliferation (PMID: 25043025, PMID: 32690037). |
| DrugClasses | CDK7 Inhibitor 16 |
| CAS Registry Number | 1604810-83-4 |
| NCIT ID | NA |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Fulvestrant + THZ1 | Fulvestrant THZ1 | 0 | 0 |
| Olaparib + THZ1 | Olaparib THZ1 | 0 | 0 |
| THZ1 | THZ1 | 1 | 0 |