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| Drug Name | OTS167 |
| Trade Name | |
| Synonyms | OTSSP167 |
| Drug Descriptions |
OTS167 is a selective inhibitor of maternal embryonic leucine zipper kinase (MELK), which can lead to anti-tumor activity (PMID: 26918358, PMID: 30061363). |
| DrugClasses | |
| CAS Registry Number | 1431698-10-0 |
| NCIT ID | C11156 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Camptothecin + OTS167 | Camptothecin OTS167 | 0 | 0 |
| Gilteritinib + OTS167 | Gilteritinib OTS167 | 1 | 0 |
| OTS167 | OTS167 | 1 | 3 |