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Drug Name | Mobocertinib |
Trade Name | Exkivity |
Synonyms | TAK-788|TAK788|AP32788|AP-32788|AP 32788 |
Drug Descriptions |
Exkivity (mobocertinib) inhibits EGFR and ERBB2 (HER2), with selectivity for mutant forms including EGFR exon 20 insertions, potentially resulting in growth inhibition in EGFR or ERBB2-mutant cancer cells (PMID: 33632775). |
DrugClasses | EGFR Exon 20 Insertion Inhibitor 15 EGFR Inhibitor (Pan) 63 HER2 Inhibitor 44 |
CAS Registry Number | 1847461-43-1 |
NCIT ID | C126752 |