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| Drug Name | SRA737 |
| Trade Name | |
| Synonyms | CCT245737|CCT-245737 |
| Drug Descriptions |
SRA737 (CCT245737) is a selective oral inhibitor of CHK1, which may enhance sensitivity of tumor cells to chemotherapeutics, thereby resulting in increased antitumor activity (PMID: 27167172, PMID: 31470128). |
| DrugClasses | CHK1 Inhibitor 18 |
| CAS Registry Number | 1489389-18-5 |
| NCIT ID | C129580 |
| Therapy Name | Drugs | Efficacy Evidence | Clinical Trials |
|---|---|---|---|
| Gemcitabine + SRA737 | Gemcitabine SRA737 | 0 | 0 |
| SRA737 | SRA737 | 0 | 0 |
| SRA737 + STP-B | SRA737 STP-B | 0 | 0 |